综合无码一区二区三区四区五区丨国产成人一区二区三区视频免费丨国产熟睡乱子伦视频观看软件丨亚洲av乱码一区二区三区观影丨2022国产精品自拍

Cat#：215P13
序列（三字母）：Myristoyl-His-Ser-Asp-Ala-Val-Phe-Thr-Asp-Asn-Tyr-Thr-Lys-Leu-Arg-Lys-Gln-Met-Ala-Val-Lys-Lys-Tyr-Leu-Asn-Ser-Ile-Lys-Lys-Gly-Gly-Thr-OH trifluoroacetate salt
序列（單字母）：Myristoyl-HSDAVFTDNYTKLRKQMAVKKYLNSIKKGGT
類似名：PG 99-465
分子式：C???H???N??O??S
分子量：3753.47
合成方法：Synthetic
存儲條件：-20 ± 5 °C
應用：Cancer Research
描述：PG 99-465 is a high affinity, selective VPAC2 receptor antagonist. It exhibited a 100-fold preference for the VPAC2 over the VPAC1 receptor. The compound showed partial agonistic activity on the VPAC1 receptor and was inactive on the VPAC2 receptor transfected in CHO cells, as well as on naturally expressed human VPAC2 receptors in the SUP T1 cell line. Dickson et al. observed an agonistic effect of PG99-465 on the human VPAC1 and PAC1 receptors. When applied singly, PG99-465 increased [cAMP](i) at all three hVPAC/PAC receptor subtypes.